Process for the synthesis of substituted piperazinones via Mitsu

Organic compounds -- part of the class 532-570 series – Organic compounds – Nitrogen attached directly or indirectly to the purine ring...

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544384, C07D40106, C07D24108

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active

061601187

ABSTRACT:
The present invention is directed to a process for synthesizing substituted piperazinones, which are useful intermediates for making farnesyl-protein transferase inhibitors, using a Mitsunobu reaction.

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