Process for the removal of exocyclic base protecting groups

Organic compounds -- part of the class 532-570 series – Organic compounds – Carbohydrates or derivatives

Reexamination Certificate

Rate now

  [ 0.00 ] – not rated yet Voters 0   Comments 0

Details

Reexamination Certificate

active

07872121

ABSTRACT:
Nitrogen-protecting groups are removed from the exocyclic nucleobase portion of a 2′-O protected nucleotide or 2′-halo nucleotide by contacting the nucleotide with an inorganic base. Typical is the removal of t-butylphenoxyacetyl protecting groups from the nucleobase portion of a 2′-O protected nucleotide on which the 2′-O protecting group is t-butyldimethylsilyl, removal or deprotection being accomplished by contact with a potassium carbonate solution.

REFERENCES:
patent: 5552539 (1996-09-01), Duplaa et al.
patent: 5808039 (1998-09-01), Reddy et al.
patent: 6664388 (2003-12-01), Nelson
(R) Schnetz-Boutaud et al., “Synthesis of Oligonucleotides Containing the Alkali-Labile Pyrimidopurinone Adduct, M1G,” Chemical Research in Toxicology, 13(2), 90-95 (2000).
(S) Fujimoto et al., “Synthesis and Cleavage of Oligonucleotides Containing a 5-Hydroxyuracil Residue in a Defined State,” Chemical Research in Toxicology, 10(11), 1254-1258 (1997).
N. D. Sinha et al, Labile Exocyclic Amine Protection (etc.), Biochimie, 1993, pp. 13-23, vol. 75, Elsevier, Paris.

LandOfFree

Say what you really think

Search LandOfFree.com for the USA inventors and patents. Rate them and share your experience with other people.

Rating

Process for the removal of exocyclic base protecting groups does not yet have a rating. At this time, there are no reviews or comments for this patent.

If you have personal experience with Process for the removal of exocyclic base protecting groups, we encourage you to share that experience with our LandOfFree.com community. Your opinion is very important and Process for the removal of exocyclic base protecting groups will most certainly appreciate the feedback.

Rate now

     

Profile ID: LFUS-PAI-O-2675101

  Search
All data on this website is collected from public sources. Our data reflects the most accurate information available at the time of publication.