Process for the racemization of...

Details Process for the racemization of... Process for the racemization of...

2005-09-27

2005-09-27

Chang, Celia (Department: 1625)

Organic compounds -- part of the class 532-570 series

Organic compounds

Heterocyclic carbon compounds containing a hetero ring...

C546S240000

Reexamination Certificate

active

06949650

ABSTRACT:
A process for the racemization of enantiomerically enriched 1-benzyl-4-(4-fluorophenyl)-3-hydroxymethyl-1,2,3,6-tetrahydropyridine which is a useful intermediate in the preparation of paroxetine. Formula (A) means that the compound (I) has an enantiomeric excess of one enantiomer over the other enantiomer. R1and R2are defined as in claim1.

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