Organic compounds -- part of the class 532-570 series – Organic compounds – Nitrogen attached directly or indirectly to the purine ring...
Patent
1995-06-02
1997-04-29
Ford, John M.
Organic compounds -- part of the class 532-570 series
Organic compounds
Nitrogen attached directly or indirectly to the purine ring...
5482646, 5482632, C07D40310
Patent
active
056250649
ABSTRACT:
Described is a process for preparing triazolone compounds of the formula ##STR1## comprising heating a mixture of a compound of the formula ##STR2## and a hydrazine derivative of the formula R.sup.5 --NH--NH--CHO, R.sup.5 --NH--NH--C(O)OC(CH.sub.3).sub.3 or R.sup.5 --NH--NH--C(O)OCH.sub.2 C.sub.6 H.sub.5, optionally in the presence of an added base.
REFERENCES:
patent: 4028344 (1977-06-01), Lange et al.
patent: 4619931 (1986-10-01), Heeres et al.
patent: 4735942 (1988-04-01), Heeres et al.
patent: 4791111 (1988-12-01), Heeres et al.
patent: 4861879 (1989-08-01), Heeres et al.
patent: 5039676 (1991-08-01), Saksena et al.
patent: 5256793 (1993-10-01), Bailey et al.
patent: 5403937 (1995-04-01), Saksena et al.
Greene, et al., "Protective Groups in Organic Synthesis", 2 ed., pp. 10-142, John Wiley & Sons (New York, 1991).
Kobayashi, et al., Bull. Chem. Soc. Jpn., 62, 3038-3040 (1989).
Temple, Jr., et al., "Triazoles 1,2,4", The Chemistry of Heterocyclic Compounds, John Wiley & Sons, New York (1981), pp. 372-373.
Temple et al, "Triazoles 1,2,4" The Chemistry of Heterocyclic Compounds John Wiley & Sons, N.Y. (1981) pp. 457-459.
Cram & Hammond, "Organic Chemistry", 2nd Edition, McGraw Hill Book On, N.Y. (1964) pp. 565-567 & pp. 249-251 & pp. 377-379 & pp. 250-251 & pp. 351-352 .
Andrews David R.
Gala Dinesh
Gosteli Jacques
Guenter Frank
Leong William
Blasdale John
Ford John M.
Schering Corporation
LandOfFree
Process for the preparation of triazolones does not yet have a rating. At this time, there are no reviews or comments for this patent.
If you have personal experience with Process for the preparation of triazolones, we encourage you to share that experience with our LandOfFree.com community. Your opinion is very important and Process for the preparation of triazolones will most certainly appreciate the feedback.
Profile ID: LFUS-PAI-O-707040