Organic compounds -- part of the class 532-570 series – Organic compounds – Boron containing
Reexamination Certificate
2006-12-05
2006-12-05
Kumar, Shailendra (Department: 1621)
Organic compounds -- part of the class 532-570 series
Organic compounds
Boron containing
C568S006000, C562S007000, C562S444000, C562S447000, C562S448000
Reexamination Certificate
active
07145040
ABSTRACT:
The present invention provides process useful for the preparation of intermediates which are useful in the preparation of amino acids useful in preparing peptide receptor modulators, for example agonists or partial agonists of such peptide receptors. Such peptide receptor modulators include, for example glucagon like peptide-1 receptor modulators which are useful for the amelioration of the diabetic condition.
REFERENCES:
patent: 3674836 (1972-07-01), Cregar
patent: 3983140 (1976-09-01), Endo et al.
patent: 4027009 (1977-05-01), Grier et al.
patent: 4231938 (1980-11-01), Monaghan et al.
patent: 4346227 (1982-08-01), Terahara et al.
patent: 4448784 (1984-05-01), Glamkowski et al.
patent: 4450171 (1984-05-01), Hoffman et al.
patent: 4499289 (1985-02-01), Baran et al.
patent: 4613610 (1986-09-01), Wareing
patent: 4647576 (1987-03-01), Hoefle et al.
patent: 4681893 (1987-07-01), Roth
patent: 4686237 (1987-08-01), Anderson
patent: 4759923 (1988-07-01), Buntin et al.
patent: 4871721 (1989-10-01), Biller
patent: 4924024 (1990-05-01), Biller
patent: 5006530 (1991-04-01), Angerbauer et al.
patent: 5011930 (1991-04-01), Fujikawa et al.
patent: 5177080 (1993-01-01), Angerbauer et al.
patent: 5260440 (1993-11-01), Hirai et al.
patent: 5273995 (1993-12-01), Roth
patent: 5354772 (1994-10-01), Kathawala
patent: 5385929 (1995-01-01), Bjorge et al.
patent: 5488064 (1996-01-01), Sher
patent: 5491134 (1996-02-01), Sher et al.
patent: 5506219 (1996-04-01), Robl
patent: 5541204 (1996-07-01), Sher et al.
patent: 5594016 (1997-01-01), Ueno et al.
patent: 5595872 (1997-01-01), Wetterau, II et al.
patent: 5612359 (1997-03-01), Murugesan
patent: 5614492 (1997-03-01), Habener
patent: 5686104 (1997-11-01), Mills et al.
patent: 5691322 (1997-11-01), Robl
patent: 5712279 (1998-01-01), Biller et al.
patent: 5712396 (1998-01-01), Magnin et al.
patent: 5739135 (1998-04-01), Biller et al.
patent: 5753675 (1998-05-01), Wattanasin
patent: 5760246 (1998-06-01), Biller et al.
patent: 5770615 (1998-06-01), Cheng et al.
patent: 5776983 (1998-07-01), Washburn et al.
patent: 5827875 (1998-10-01), Dickson, Jr. et al.
patent: 5885983 (1999-03-01), Biller et al.
patent: 5962440 (1999-10-01), Sulsky
patent: 5998375 (1999-12-01), Thøgersen et al.
patent: 6043265 (2000-03-01), Murugesan et al.
patent: 6545029 (2003-04-01), Vaupel
patent: 6548667 (2003-04-01), Park et al.
patent: 6737417 (2004-05-01), Jo et al.
patent: 7045652 (2006-05-01), Caron et al.
patent: 2003/0195157 (2003-10-01), Natarajan et al.
patent: 2004/0127423 (2004-07-01), Natarajan et al.
patent: 0 142 146 (1985-05-01), None
patent: 0 221 025 (1987-05-01), None
patent: 2 596 393 (1987-10-01), None
patent: 2 205 837 (1988-12-01), None
patent: WO 86/03488 (1986-06-01), None
patent: WO 86/07054 (1986-12-01), None
patent: WO 96/38144 (1996-12-01), None
patent: WO 97/12613 (1997-04-01), None
patent: WO 97/12615 (1997-04-01), None
patent: WO 97/21993 (1997-06-01), None
patent: WO 99/00353 (1999-01-01), None
patent: WO 99/38501 (1999-08-01), None
patent: WO 99/46272 (1999-09-01), None
patent: WO 99/61431 (1999-12-01), None
patent: WO 99/67278 (1999-12-01), None
patent: WO 99/67279 (1999-12-01), None
patent: WO 00/01389 (2000-01-01), None
U.S. Appl. No. 11/170,968, filed Jun. 30, 2005, Ewing et al.
Ashworth, D.M. et al., “2-Cyanopyrrolidides as Potent, Stable Inhibitors of Dipeptidyl Peptidase IV”, Bioorganic & Medical Chemistry Letters, vol. 6, No. 10, pp. 1163-1166 (1996).
Ashworth, D.M. et al., “4-Cyanothiazolidides as Very Potent, Stable Inhibitors of Dipeptidyl Peptidase IV”, Bioorganic & Medicinal Chemistry Letters, vol. 6, No. 22, pp. 2745-2748 (1996).
Atherton, E. et al., Chapter 1: “The Fluorenylmethoxycarbonyl Amino Protecting Group”, The Peptides: Analysis, Synthesis, Biology, vol. 9: Special Methods in Peptide Synthesis, Part C, Academic Press, Inc., publ., Udenfriend, S. et al., eds. pp. 1-38 (1987).
Barany, G. et al., Chapter 1: “Solid-Phase Peptide Synthesis”, The Peptides: Analysis, Synthesis, Biology, vol. 2: Special Methods in Peptide Synthesis, Part A, Acdemic Press, Inc., publ. Gross, E. et al., eds., pp. 1-284 (1979).
Biller, S.A. et al., “Isoprenoid (Phosphinylmethyl)phosphonates as Inhibitors of Squalene Synthetase”, Journal of Medicinal Chemistry, vol. 31, No. 10, pp. 1869-1871 (1988).
Biller, S.A. et al., “Squalene Synthase Inhibitors”, Current Pharmaceutical Design, vol. 2, No. 1, pp. 1-40 (1996).
Burgess, K. et al., “Solid Phase Syntheses of Oligoureas”, J. Am. Chem. Soc., vol. 119, No. 7, pp. 1556-1564 (1997).
Byrne, M.M. et al., “Inhibitory effects of hyperglycaemia on fed jejunal motility: potential role of hyperinsulineamia”, European Journal of Clinical Investigation, vol. 28, pp. 72-78 (1998).
Capson, T.L., “Synthesis and Evaluation of Ammonium Analogs of Carbocationic Intermediates in Squalence Biosynthesis”, dissertation, Department of Medicinal Chemistry, University of Utah, pp. iv-v, Table of Contents, 16-17, 40-43, 48-51, Summary (Jun. 1987).
Corey, E.J. et al., “Application of Unreative Analogs of Terpenoid Pyrophosphates to Studies of Multistep Biosynthesis. Demonstration That ‘Presqualene Pyrophosphate’ Is an Essential Intermediate on the Path to Squalene”, Journal of the American Chemical Society, vol. 98, No. 5, pp. 1291-1293 (1976).
Cornicelli, J.A. et al., “15-Lipoxygenase and Its Inhibition: A Novel Therapeutic Target for Vascular Disease”, Current Pharmaceutical Design, vol. 5, No. 1, pp. 11-20 (1999).
Davern, P. et al., “Chemical and Biological Reactivity of Sulfamidopenicillins”, J. Chem. Soc. Perkin Trans. 2, pp. 381-387 (1994).
Fehder, W.P. et al., “Development and Evaluation of a Chromatographic Procedure for Partial Purification of Substance P with Quantitation by an Enzyme Immunoassay”, Clinical and Diagnositc Laboratory Immunology, vol. 5, No. 3, pp. 303-307 (1998).
Fehrentz, J.-A. et al., “An Efficient Synthesis of Optically Active α-(t-Butoxycarbonylamino)-aldehydes from α-Amino Acids”, Synthesis, pp. 676-678 (1983).
Fingl, E. et al., Section I: “Introduction”, Chapter I: “General Principles”, The Pharmacological Basics of Therapeutics, 5thEd., Macmillan Publishing Co., Inc., publ., Goodman, L.S. et al., eds., pp. 1-46 (1975).
Flint, A. et al., “Glucagon-like Peptide 1 Promotes Satiety and Suppresses Energy Intake in Humans”, J. Clin. Invest., vol. 101, No. 3, pp. 515-520 (1998).
Gennaro, A.R., ed., Remington's Pharmaceutical Sciences, 18thEd., Mack Publishing Company, publ., pp. xv-xvi (table of contents) (1990).
Gennaro, A.R., ed., Remington: Practice of the Science and Pharmacy, 19thEd., Mack Publishing Company, publ., pp. xv-xvi (table of contents) (1995).
Gennaro, A.R., ed., Remington: Practice of the Science and Pharmacy, vol. II, 19thEd., Mack Publishing Company, publ., pp. vii-viii (table of contents) (1995).
Ghiselli, G., “The Pharmacological Profile of FCE 27677: A Novel ACAT Inhibitor with Potent Hypolipidemic Activity Mediated by Selective Suppression of the Hepatic Secretion of ApoB-100-Containing Lipoprotein”, Cardiovascular Drug Reviews, vol. 16, No. 1, pp. 16-30 (1998).
Gluschankof, P. et al., “Enzymes processing somatostatin precursors: An Arg-Lys esteropeptidase from the rat brain cortex converting somatostatin-28 into somatostatin-14”, Proc. Natl. Acad. Sci. USA, vol. 81, pp. 6662-6666 (1984).
Gutzwiller, J.-P. et al., “Glucagon-like peptide-1: a potent regulator of food intake in humans”, Gut, vol. 44, pp. 81-86 (1999).
Hara, S. “Ileal Na+/bile acid cotrasporter inhibitors”, Drugs of the Future, vol. 24, No. 4, pp. 425-430 (1999).
Holst, J.J., “Glucagon-like Peptide-1, A Gastrointestinal Hormone with a Pharmaceutical Potential”, Current Medicinal Chemistry, vol. 6, No. 11, pp. 1005-1017 (1999).
Ito, Y. et al., “Difference in cholesterol-bin
Kumar K. Selva
Mathur Arvind
Bergen Briana C.
Bristol-Myers Squibb Co.
Carey Brian C.
Kumar Shailendra
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