Process for the preparation of 1,3-substituted indenes and...

Details Process for the preparation of 1,3-substituted indenes and... Process for the preparation of 1,3-substituted indenes and...

2007-03-06

2007-03-06

Crane, L. E. (Department: 1623)

Chemistry of hydrocarbon compounds

Compound or reaction product mixture

Aromatic

C585S269000, C585S419000, C558S303000, C558S311000, C560S018000, C560S155000

Reexamination Certificate

active

11286055

ABSTRACT:
The present invention relates to processes for the preparation of any of the intermediate 1,3-substituted indenes of the formulae (Ia), (Ib) and (Ic) or a mixture thereof:wherein R1, R2, R3, R4, and R5are defined herein. Compounds of formulae (Ia), (Ib) and (Ic) or mixtures thereof are useful in the preparation of compounds of formula (II):wherein R2, R3and R6are also defined herein.

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[R] Mazzochi et al., “Synthesis and Pharmacological Activity of 2,3,4,5-Tetrahydro-1,5-methano-1H-3-benzazepines,” Journal of Medicinal Chemistry, 22(4), 455-457 (Apr. 1979).
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