Drug – bio-affecting and body treating compositions – Designated organic active ingredient containing – Having -c- – wherein x is chalcogen – bonded directly to...
Patent
1998-02-17
1999-12-14
Kight, John
Drug, bio-affecting and body treating compositions
Designated organic active ingredient containing
Having -c-, wherein x is chalcogen, bonded directly to...
546 62, 546 77, 546 78, A61K 3147, C07D47102
Patent
active
060018461
ABSTRACT:
A method for preparing 1,2-dihydroquinolines that is more flexible than the Skraup reaction is provided. The method comprises treating an ortho-alkenyl aniline with a ketone in the presence of a Lewis acid. Novel intermediates and products of this method useful as steroid receptor modulators, as well as pharmaceutical compositions and methods of use thereof are also claimed.
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Carreira Erick M.
Edwards James P.
Jones Todd K.
Riggenberg Josef D.
Aulakh Charanjit S.
Elmer James Scott
Kight John
Ligand Pharmaceuticals Incorporated
Respess William L.
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