Process for producing optically active phosphorus...

Organic compounds -- part of the class 532-570 series – Organic compounds – Phosphorus containing

Reexamination Certificate

Rate now

  [ 0.00 ] – not rated yet Voters 0   Comments 0

Details

Reexamination Certificate

active

07411096

ABSTRACT:
The present invention provides a process for producing an optically active phosphorus heterocyclic dimer including reacting, in the presence of a base, primary phosphine represented by formula (1)in-line-formulae description="In-line Formulae" end="lead"?R—PH2  (1)in-line-formulae description="In-line Formulae" end="tail"?is reacted with a compound represented by formula (2)in-line-formulae description="In-line Formulae" end="lead"?Y—CnH2n—Y  (2)in-line-formulae description="In-line Formulae" end="tail"?in the presence of a base; the product is reacted with boron trihydride, oxygen, or sulfur to obtain a phosphorus heterocyclic compound represented by formula (3):the resultant compound is dimerized to produce a phosphorus heterocyclic dimer represented by formula (4):and then oxygen, sulfur, or borane is removed from the resultant phosphorus heterocyclic dimer to obtain an optically active phosphorus heterocyclic dimer represented by formula (5):

REFERENCES:
patent: 7169953 (2007-01-01), Zhang et al.
patent: WO 03/042135 (2003-05-01), None
Ohashi et al. (Heterocycles 2000, 52(2), 905-910)—a printout of the CAS Abstract and reacation are attached.
Burk, J. et al., “Preparation and Use of C2-Symmetric Bis(phospholanes): Production of α-Amino Acid Derivatives via Highly Enantioselective Hydrogenation Reactions”, J. Am. Chem. Soc., 1993, pp. 10125-10138, vol. 115, No. 22, American Chemical Society.
Imamoto, T. et al., “P-Chiral Bis(trialkylphosphine) Ligands and Their Use in Highly Enantioselective Hydrogenation Reactions”, J. Am. Chem. Soc., 1998, pp. 1635-1636, vol. 120, No. 7, American Chemical Society.
Imamoto T. et al., “Optically Active 1,1′-Di-tert-butyl-2,2′-diphosphetanyl and Its Application in Rhodium-Catalyzed Asymmetric Hydrogenations”, Synthesis 2004, 2004, pp. 1353-1358, No. 9, Georg Thieme Verlag Stuttgart, New York.

LandOfFree

Say what you really think

Search LandOfFree.com for the USA inventors and patents. Rate them and share your experience with other people.

Rating

Process for producing optically active phosphorus... does not yet have a rating. At this time, there are no reviews or comments for this patent.

If you have personal experience with Process for producing optically active phosphorus..., we encourage you to share that experience with our LandOfFree.com community. Your opinion is very important and Process for producing optically active phosphorus... will most certainly appreciate the feedback.

Rate now

     

Profile ID: LFUS-PAI-O-4012630

  Search
All data on this website is collected from public sources. Our data reflects the most accurate information available at the time of publication.