Process for preparing the antiviral agent [1S-(1alpha,3...

Organic compounds -- part of the class 532-570 series – Organic compounds – Four or more ring nitrogens in the bicyclo ring system

Reexamination Certificate

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C544S276000, C548S215000, C556S436000, C556S441000, C556S473000, C556S465000, C556S413000, C556S443000, C556S482000, C556S489000, C562S126000, C568S660000

Reexamination Certificate

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07034152

ABSTRACT:
Processes are disclosed for preparing the antiviral agent entecavir. A resin adsorption process for the isolation and purification of entecavir is also disclosed. Various intermediates useful in the preparation of entecavir are also disclosed.

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