Organic compounds -- part of the class 532-570 series – Organic compounds – Four or more ring nitrogens in the bicyclo ring system
Patent
1981-12-28
1984-03-06
Waltz, Thomas A.
Organic compounds -- part of the class 532-570 series
Organic compounds
Four or more ring nitrogens in the bicyclo ring system
546143, 546146, 548127, 548128, 548135, 548140, 548163, 548167, 548337, 548341, 560 34, 564 47, 564 48, 564 50, 564 52, 564 53, 564 54, 564 55, 564 56, 564 57, 564 59, 564 60, 564 61, C07C12700, C07C12715, C07C12717, C07C12719
Patent
active
044355670
ABSTRACT:
A process for the preparation of substituted urea derivatives, and compositions and concentrates for the same purpose are disclosed. According to the process the substituted urea derivatives of formula (I) ##STR1## wherein R is hydrogen, alkyl, aryl, cycloalkyl or aralkyl, R.sup.1 and R.sup.2 are hydrogen, alkyl, alkenyl, alkinyl, alkoxy, oxyalkyl, cycloalkyl, aralkyl, alkoxycarbonylalkyl, aryl or heteroaryl, or R.sup.1 and R.sup.2 together with the adjacent nitrogen atom may form a saturated or unsaturated heterocycle, or a condensed and/or substituted ring system, and said heterocycle or said condensed and/or substituted ring system may contain also a sulfo group,
can be manufactured by reacting an amine of formula (II) ##STR2## with an N-carbamoyl-benzoic acid sulfimide derivative of formula (III) ##STR3## The disclosed N-acylating composition comprises of from 3 to 60% by weight, preferably of from 5 to 50% by weight sulfimide derivative of formula (III), of from 97 to 40% by weight, preferably of from 95 to 50% by weight solvent, and if desired, an organic or inorganic base.
The disclosed N-acylating concentrate comprises of from 60 to 95.5% by weight N-acylating agent of formula (III) and of from 4.5 to 40% by weight additives.
REFERENCES:
Theilheimer, Synthetic Methods of Organic Chemistry, vol. 16, #434, Basel-Karger Publishers, N.Y., N.Y.
Shioyama et al., CA78: 124577y (1973).
McClelland et al., CA 42: 907h (1947).
Klyuev et al., CA 71: 22053n (1969).
Bodnar Janos
Lugosi Gyorgy
Simandi Laszlo
Simay Antal
Somfai Eva
Chinoin Gyogyszer es Vesgyeszeti Termekek Gyara R. T.
Dubno Herbert
Ross Karl F.
Waltz Thomas A.
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