Process for preparing substituted polyazamacrocycles

Organic compounds -- part of the class 532-570 series – Organic compounds – Unsubstituted hydrocarbyl chain between the ring and the -c-...

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540451, 540452, C07D22502

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active

057213615

ABSTRACT:
A process for preparing a substituted polyazamacrocycle is provided which comprises contacting a diamine or triamine and a dicarboxylic acid or ester or anhydride thereof in the presence of a suitable base and a suitable solvent to produce the substituted polyazamacrocycle provided that when an ester of said dicarboxylic acid is used, said suitable base is optional, and when said dicarboxylic acid or an anhydride of said dicarboxylic acid is used, the reaction mixture further comprises a suitable coupling agent.

REFERENCES:
patent: 4569750 (1986-02-01), Brownswell et al.
patent: 4923985 (1990-05-01), Gansow et al.
patent: 5126464 (1992-06-01), Burrows et al.
patent: 5298618 (1994-03-01), Speranza et al.
patent: 5322681 (1994-06-01), Klaveness
patent: 5324334 (1994-06-01), Brois et al.
patent: 5386028 (1995-01-01), Tilstam et al.
Dariez et al., Tetra Letters., vol. 48, No. 21, pp. 4347-4358, 1992.
Fieser & Fieser., Reapents for Org. Synthesis p. 1313, 1967.
Shakir et al., Tetrahedron., vol. 56, pp. 3339-3344, 1991.
Jean-Paul Behr et al. Macrotricyclic and Macropentacyclic Ditopic Receptor Molecules, Synthesis, Crystal Structure and Substrate Binding, Tetrahedron Letters, vol. 28, No. 18, pp. 1989-1992, (1987).
Marie-Christine Duriez et al. Macrocylic Polyether Tetralactams I: Synthesis and Cyclization Studies, Tetrahedron, vol. 48, No. 21, pp. 4347-4358 (1992).
Louis F. Fieser et al. Reagents for Organic Synthesis, John Wiley and Sons, Inc. (1967).
Krzysztof E. Krakowiak et al. Synthesis of Aza-Crown Ethers, Chemical Reviews, vol. 89, No. 4, 929-972 (1989).
McMurry et al. Convenient Synthesis of Bifunctional Tetraaza Macrocycles, Bioconjugate Chem, vol. 3, No. 2, pp. 108-117, (1992).
Moberg et al. Synthesis and Structure of Macrocyclic Amides Containing a 2,2'-Dipyridylmethane Unit. A New Class of Chiral Macrocyclic Ligands, J. Org. Chem., vol. 56, pp. 3339-3344, (1991).
Mohammad Shakir et al. Divalent Cobalt, Nickel, Copper and Zinc Complexes of Tetraaza Macrocycles Bearing Polyamide Groups: Synthesis and Characterization, Tetrahedron, vol. 12, No. 23, pp. 2775-2780 (1993).

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