Process for preparing protease inhibitor intermediates

Details Process for preparing protease inhibitor intermediates Process for preparing protease inhibitor intermediates

2006-12-05

2006-12-05

Solola, Taofiq (Department: 1626)

Organic compounds -- part of the class 532-570 series

Organic compounds

Heterocyclic carbon compounds containing a hetero ring...

Reexamination Certificate

active

07145024

ABSTRACT:
The present invention includes a method for preparing cyclic alcohols. The method includes a reduction, deprotection, and rearrangement scheme. The present invention further provides a method of preparation of an intermediate useful in the synthesis of compounds that function as inhibitors of the aspartyl protease enzyme of human immunodeficiency virus (HIV).

REFERENCES:
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PCT Written Opinion.

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