Process for preparing Nebivolol

Details Process for preparing Nebivolol Process for preparing Nebivolol

2011-08-23

2011-08-23

Dentz, Bernard (Department: 1622)

Organic compounds -- part of the class 532-570 series

Organic compounds

Heterocyclic carbon compounds containing a hetero ring...

C549S398000, C549S401000

Reexamination Certificate

active

08003810

ABSTRACT:
The present invention relates to a process for preparing Nebivolol and, more particularly, to an improved process for synthesizing enantiomerically enriched 6-fluoro chroman alcohol or epoxide derivatives of formula, wherein R and X is defined in the description; as useful intermediates in the preparation of Nebivolol.

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