Organic compounds -- part of the class 532-570 series – Organic compounds – Unsubstituted hydrocarbyl chain between the ring and the -c-...
Patent
1995-05-22
1997-06-10
Grumbling, Matthew V.
Organic compounds -- part of the class 532-570 series
Organic compounds
Unsubstituted hydrocarbyl chain between the ring and the -c-...
544111, 544114, 544121, 544122, 544124, 544129, 544132, 544133, 544134, 544137, 544139, 544140, 544141, 544143, 544148, 544153, 544174, C07D41302, C07D26528, C07D26530, C07D26534
Patent
active
056376995
ABSTRACT:
Substituted heterocycles of the general structural formula: ##STR1## are tachykinin receptor antagonists useful in the treatment of inflammatory diseases, pain or migraine, asthma and emesis, and calcium channel blockers useful in the treatment of cardiovascular conditions such as angina, hypertension or ischemia.
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Chambers Mark S.
Dorn Conrad P.
Finke Paul E.
Hale Jeffrey J.
Harrison Timothy
Grumbling Matthew V.
Merck & Co. , Inc.
Rose David L.
Thies J. Eric
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