Process for preparing halogenated 2,3-O-cyclocytidine derivative

Details Process for preparing halogenated 2,3-O-cyclocytidine derivative Process for preparing halogenated 2,3-O-cyclocytidine derivative

1995-06-06

1997-01-21

Kunz, Gary L.

Organic compounds -- part of the class 532-570 series

Organic compounds

Carbohydrates or derivatives

536 2852, C07H 100, C07H 1909

Patent

active

055960936

ABSTRACT:
A process from preparing 5-halogenated 2,3-O-cyclocytidine derivatives comprising reacting 2,3-O-cyclocytidine with a halogenating reagent, preferably N-bromosuccinimide, in the presence of an acid such as acetic or trifluoroacetic.

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