Process for preparing benzo[b]thiophenes

Details Process for preparing benzo[b]thiophenes Process for preparing benzo[b]thiophenes

1998-04-29

1999-11-30

Chang, Ceila

Organic compounds -- part of the class 532-570 series

Organic compounds

Heterocyclic carbon compounds containing a hetero ring...

540536, 548525, C07D40912

Patent

active

059945478

ABSTRACT:
The preparation of benzo[b]thiophenes by the acylation of alkoxy protected starting materials followed by demethylation using essentially odorless thiol compounds are provided herewith. Demethylation may be carried out in the same reaction vessel without isolation of the acylated, protected material.

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