Process for preparing 6-[(isoxazolinyl)methyl]penicillanic acid

Details Process for preparing 6-[(isoxazolinyl)methyl]penicillanic acid Process for preparing 6-[(isoxazolinyl)methyl]penicillanic acid

1994-02-07

1996-01-30

Rizzo, Nicholas

Organic compounds -- part of the class 532-570 series

Organic compounds

Heterocyclic carbon compounds containing a hetero ring...

C07D49900, A61K 3143

Patent

active

054881064

ABSTRACT:
The invention provides a novel class of 6-(isoxazolinyl)methyl penicillanic acid 1,1-dioxide compounds having the formula: ##STR1## wherein M, X, R.sup.2, R.sup.3, R.sup.4 and R.sup.5 are described in the specification;

REFERENCES:
patent: 5015473 (1991-05-01), Chen
T. Greene, Protective Groups in Organic Synthesis, J. Wiley & Sons, 1981, pp. 53-61.
Volkmann et al., J. Org. Chem., vol. 47, pp. 33-44 (1982).
Hannessian, Tetrahedron, vol. 45, pp. 941-950 (1989).
N. A. Kuck, et al., "Antibiotic Agents and Chemotherapy", vol. 33, 1989, pp. 1964-1969.
A. Brandi et al., J. Org. Chem., vol. 54, pp. 3073-3077 (1989).
Mukaiyama et al., J. Am. Chem. Soc., vol. 82, pp. 5339-5345 (1960).
Weeks and Volkmann, Tetrahedron Letters, vol. 27, pp. 1549-1552 (1986).
L. A. Reed et al., Tetrahedron Letters, vol. 28, 3431-3434 (1987).
Hannessian et al., Tetrahedron Letters, vol. 27, pp. 4857-4860 (1986).
Kou-Chang Liu et al., J. Org. Chem., vol. 45, pp. 3916-3918 (1980).
Just et al., J. Org. Chem., 52, 36-59 (1987).
Foulds et al., J. Chem. Soc. Perkin Trans I, 963-968 (1985).
D. M. Vyas et al., Tetrahedron Letters, 25, 487-490 (1984).
H. C. New, "Antibiotic Inhibitors of Bacterial Cell Wall Biosynthesis", D. J. Tipper ed, Pergamon Press, 1987, 241-259.
K. Bush, "Antibiotic Agents and Chemotherapy", vol. 33, 1989, pp. 259-276.
Yang et al., "Antibiotic Agents and Chemotherapy", vol. 36, 1992, 1155-1157.

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