Process for preparing 2-methyl-thieno-benzodiazepine

Details Process for preparing 2-methyl-thieno-benzodiazepine Process for preparing 2-methyl-thieno-benzodiazepine

2008-01-22

2008-01-22

Coleman, Brenda (Department: 1624)

Drug, bio-affecting and body treating compositions

Designated organic active ingredient containing

Heterocyclic carbon compounds containing a hetero ring...

C540S557000

Reissue Patent

active

10023132

ABSTRACT:
2-Methyl-4-(4-methyl-1-piperazinyl)-10H-thieno-[2,3-b][1,5]benzodiazepine, or an acid salt thereof, has pharmaceutical properties, and is of particular use in the treatment of disorders of the central nervous system. The compound has the following structure:

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DRL Corrected Conclusion of Law, Mar. 24, 2004.
DRL Corrected Findings of Fact, Mar. 24, 2004.
DRL Corrected Post -Trial Brief, Mar. 24, 2004.
DRL Reply Brief Dec. 10, 2005.
DRL Appeal Brief Aug. 15, 2005.
Lilly v Zenith Goldline-CAFC Dec. 26, 2006.
Lilly's CoL, Apr. 21, 2004.
Lilly's Counter FoF CoL, Apr. 21, 2004.
Lilly's FoF, Apr. 21, 2004.
Lilly's Post-Trial Brief, Apr. 21, 2004.
Lilly's Supplemental Brief, May 7, 2004.
Zenith Post-Trial Brief, Mar. 22, 2004.
Zenith Appeal Brief Aug. 15, 2005.
Zenith Reply Brief, Mar. 22, 2004.
Zenith Reply to Lilly's CoL, May 12, 2004.

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