Organic compounds -- part of the class 532-570 series – Organic compounds – Nitrogen attached directly or indirectly to the purine ring...
Patent
1997-09-16
1999-01-19
Bernhardt, Emily
Organic compounds -- part of the class 532-570 series
Organic compounds
Nitrogen attached directly or indirectly to the purine ring...
544368, 544374, C07D24104
Patent
active
058615121
ABSTRACT:
Intermediates of structural formula ##STR1## can be made by reacting a primary or secondary amine with glycosidol or an activated derivative thereof. The process and intermediates are useful for synthesizing HIV protease inhibitor compounds.
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Chemical Abstracts. vol. 86, 1997 p. 89161, Section 86: 89157c, Reinhold et al.
Askin David
Reider Paul
Rossen Kai
Varsolona Richard J.
Volante Ralph P.
Bernhardt Emily
Merck & Co. , Inc.
Walton Kenneth R.
Winokur Melvin
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