Process for fluorinating 1-phenyl-2-amino-1,3-propanediol compou

Details Process for fluorinating 1-phenyl-2-amino-1,3-propanediol compou Process for fluorinating 1-phenyl-2-amino-1,3-propanediol compou

1993-05-24

1994-07-26

Daus, Donald G.

Organic compounds -- part of the class 532-570 series

Organic compounds

Heterocyclic carbon compounds containing a hetero ring...

548237, C07D26310

Patent

active

053328353

ABSTRACT:
Replacement with fluorine of the primary hydroxy group of 1-phenyl-2-amino-1,3-propanediol compounds wherein the secundary hydroxy group and the amino group have been suitably protected.
The reaction is carried out with an inorganic fluoride in a polyglycol.
New oxazoline compounds particularly useful in said-process.

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