Organic compounds -- part of the class 532-570 series – Organic compounds – Heterocyclic carbon compounds containing a hetero ring...
Patent
1991-11-27
1994-11-15
Cintins, Marianne M.
Organic compounds -- part of the class 532-570 series
Organic compounds
Heterocyclic carbon compounds containing a hetero ring...
546284, 546304, 546309, 546312, C07D21374, C07D21156
Patent
active
053649435
ABSTRACT:
Substituted piperidines and related compounds of the formula ##STR1## wherein R.sup.1 and R.sup.2 are herein defined are disclosed.
REFERENCES:
patent: 3560510 (1971-02-01), Warawa et al.
patent: 4358446 (1982-11-01), Haken et al.
patent: 4552960 (1985-11-01), Krumkalns et al.
patent: 4680283 (1987-07-01), Veber et al.
patent: 5138060 (1992-08-01), Godek et al.
patent: 5162339 (1992-11-01), Lowe
Dickinson et al., "Thromboxane Synthetase Inhibitors and Antagonists", vol. 22 Annual Reports in Medicinal Chemistry, 95-105 (1987).
E. J. Warawa et al. "Quinuclidine Chemistry", J. Med. Chem., 18, 587 (1975).
Sandberg et al. "Substance P," J. Med. Chem., 25, 1009, (1982).
P. J. Goadsby et al. "Release of Vasoactive Peptides" Ann. Neurol., 23, 193 (1988).
Regoli, "Neurokinin Agonists & Antagonists" Elsevier Scientific Publishers, Amsterdam, pp. 85-95 (1987).
L. S. Trifonov et al. "Synthesis of 1,2-Five-Ring-Annellated Barrelenes" Helvetica Chimica Acta, 70, 4, 1732-1736 (1987).
A. S. Yanni et al., "Synthesis & biological Activity" Indian J. Chem., 21B (7), 705-6, (1982).
Y. P. Gupta et al. "Synthesis of 2,12-Diazachrysene via Benzyne Cyclization Reaction," Indian J. Chem., 19B (5), 400-1, (1980).
V. N. Gogte et al. "Infrated Spectral Study of the Effect of Substitution on Conformation and Hydrogen Bonding in 3-(aryl-amino)propanols," Indian J. Chem., 17B (3), 230-2, (1979).
S. V. Kessar et al. "New Routes to Condensed Polynuclear Compounds," Tetrahedron, 29, Pergamon Press, (GB), 419-424, 1978.
G. N. Walker et al. "Synthesis of Caried Heterocyclic & Substituted Arylalkyl" J. Med. Chem., 9, No. 4, (1966), 624-630.
G. N. Walker et al. "Application of Sodium Borohydride" Journal of Organic Chemistry, 26, No. 8, (1961), American Chemical Society, (US), 2740-2747.
Suman Rakhit et al. "Formation of Animals from Amines via Pummerer Rearrangement," Can. J. Chem., 57, No. 10, 1153 (1979).
Godek Dennis M.
Gut Sally
Rosen Terry J.
Wint Lewin
Butterfield Garth
Cintins Marianne M.
Ginsburg Paul H.
Pfizer Inc.
Richardson Peter C.
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