Preparation of Anilineboronic acids and derivatives thereof

Details Preparation of Anilineboronic acids and derivatives thereof Preparation of Anilineboronic acids and derivatives thereof

2007-03-27

2007-03-27

Davis, Brian (Department: 1621)

Organic compounds -- part of the class 532-570 series

Organic compounds

Amino nitrogen containing

C568S006000

Reexamination Certificate

active

10846463

ABSTRACT:
A process for preparing anilineboronic acid derivative of the formula I,by converting an aniline to a diprotected aniline by introducing two protecting groups, metalating the diprotected aniline with a metalating agent and simultaneously or subsequently reacting with a boronic ester B(OR1,2,3)3to form a protected anilineboronic ester, which is converted, by detaching the protecting groups, to the anilineboronic esters of the formula (I).

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