Organic compounds -- part of the class 532-570 series – Organic compounds – Heterocyclic carbon compounds containing a hetero ring...
Patent
1994-05-17
1995-08-15
Richter, Johann
Organic compounds -- part of the class 532-570 series
Organic compounds
Heterocyclic carbon compounds containing a hetero ring...
C07D48700
Patent
active
054420563
ABSTRACT:
The present invention is directed to a process of making 2-aryl carbapenems of formula 1 from a compound of formula A. ##STR1## wherein compound A is reacted with a silyl protected boronic acid compound of the formula B: ##STR2## and wherein Ar is selected from the group consisting of: ##STR3##
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DeCamp Ann E.
Grabowski Edward J. J.
Huffman Mark A.
Xavier Lyndon C.
Yasuda Nobuyoshi
Billups Richard C.
Cook Rebecca
Daniel Mark R.
DiPrima Joseph F.
Merck & Co. , Inc.
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