Practical synthesis of benzoxazinones useful as HIV reverse tran

Details Practical synthesis of benzoxazinones useful as HIV reverse tran Practical synthesis of benzoxazinones useful as HIV reverse tran

1999-06-25

2000-11-14

Raymond, Richard L.

Organic compounds -- part of the class 532-570 series

Organic compounds

Chalcogen in the nitrogen containing substituent

C07D26518

Patent

active

061472107

ABSTRACT:
The present invention describes novel methods for the synthesis of benzoxazinone compounds which are useful as human immunodeficiency virus (HIV) reverse transcriptase inhibitors. The benzoxazinone of the formula: is particularly effective in the treatment of HIV.

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