Polar-substituted hydrocarbons

Details Polar-substituted hydrocarbons Polar-substituted hydrocarbons

1999-02-22

2000-06-06

Shah, Mukund J.

Drug, bio-affecting and body treating compositions

Designated organic active ingredient containing

Phosphorus containing other than solely as part of an...

514 64, 514218, 514247, 514248, 514252, 514253, 514311, 514314, 540553, 546 13, 546 23, 546169, 544237, 544238, A61K 3165, A61K 3127, C07C32357, C07D20714, C07D21548

Patent

active

060718951

ABSTRACT:
The present invention discloses the compounds of general formula (1) ##STR1## wherein R.sup.1, R.sup.2, R.sup.3 are optionally substituted carbonyl and amide derivatives which are useful as inhibitors of retroviral proteases, and are effective in treating conditions characterized by unwanted activity of these enzymes, such as acquired immume deficiency syndrome.

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