Piperidine and azetidine derivatives as GlyT1 inhibitors

Drug – bio-affecting and body treating compositions – Designated organic active ingredient containing – Heterocyclic carbon compounds containing a hetero ring...

Reexamination Certificate

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Details

C514S318000, C514S326000

Reexamination Certificate

active

07655644

ABSTRACT:
The present invention provides compounds of formula (I), wherein both p's are one or two, R1is generally heteroaryl or cycloalkyl, R2is C3-6cycloalkyl or phenyl and R3is heteroaryl, and pharmaceutically acceptable salts thereof, as GlyT1 inhibitors for treating schizophrenia, pharmaceutical compositions comprising the same and methods for their preparation.

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patent: 2007/0105902 (2007-05-01), Lindsley et al.
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patent: WO 03/088908 (2003-10-01), None
patent: WO 2005/094514 (2005-10-01), None
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Copending U.S. Appl. No. 12/084,027, filed Oct. 27, 2006, U.S. National Stage Entry of PCT/GB06/041699, published as WO 2007/053400.
Copending U.S. Appl. No. 12/085,340, filed Nov. 23, 2006, U.S. National Stage Entry of PCT/GB06/050411, published as WO 2007/060484.

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