Phosphorylcarbamates of rapamycin and oxime derivatives thereof

Details Phosphorylcarbamates of rapamycin and oxime derivatives thereof Phosphorylcarbamates of rapamycin and oxime derivatives thereof

1993-10-08

1995-02-21

Bond, Robert T.

Organic compounds -- part of the class 532-570 series

Organic compounds

Unsubstituted hydrocarbyl chain between the ring and the -c-...

A61K 31395, C07D49106

Patent

active

053917308

ABSTRACT:
A compound of the structure ##STR1## wherein R.sup.1 and R.sup.2 are each, independently, hydrogen, or ##STR2## R.sup.3 and R.sup.4 are each, independently, hydrogen, Ar, or --(CR.sup.6 R.sup.7).sub.a Y(CR.sup.8 R.sup.9).sub.b Z, or R.sup.3 and R.sup.4 may be taken together to form a 5-7 membered ring;

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