Drug – bio-affecting and body treating compositions – Designated organic active ingredient containing – Carbohydrate doai
Patent
1998-05-06
2000-10-31
Wilson, James O.
Drug, bio-affecting and body treating compositions
Designated organic active ingredient containing
Carbohydrate doai
514 48, 514 51, 514 52, 536 267, 536 2671, 536 2672, 536 2674, 536 268, 536 269, 568 8, 568 13, 568 14, A61K 3170, A01N 4304, C07F 0902
Patent
active
061403105
ABSTRACT:
The composition and methods of synthesis of phosphorus prodrugs are described. These methods can be used to convert negatively charged phosphorus bearing drugs into neutrally charged; lipid soluble prodrugs which are able to passively diffuse into cells and into tissues in vivo. Prodrugs for a variety of antiviral and anti-leukemic agents are described.
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Drug Innovation & Design, Inc.
Wilson James O.
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