Phosphoramidite derivatives of macrocycles

Organic compounds -- part of the class 532-570 series – Organic compounds – Heterocyclic carbon compounds containing a hetero ring...

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536 171, 536 173, 536 174, 540472, C07D18722, C07F 700, C07F 96524

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active

058378669

ABSTRACT:
The invention is directed to phosphoramidite derivatives of macrocycles, such as porphyrins and expanded porphyrins, including sapphyrins and texaphyrins. The phosphoramidite derivatives are useful as intermediates in the preparation of macrocycle-oligonucleotide conjugates.

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