Organic compounds -- part of the class 532-570 series – Organic compounds – Heterocyclic carbon compounds containing a hetero ring...
Reexamination Certificate
2006-07-18
2006-07-18
Richter, Johann (Department: 1621)
Organic compounds -- part of the class 532-570 series
Organic compounds
Heterocyclic carbon compounds containing a hetero ring...
C544S402000, C544S162000, C540S609000, C546S229000
Reexamination Certificate
active
07078537
ABSTRACT:
The present invention relates to novel 1,2- or 1,3-diamine and amide compounds and pharmaceutically useful salts thereof and methods for treating central nervous system diseases. The present 1,2- or 1,3-diamine and amide compounds have high binding affinity to the sigma receptor.
REFERENCES:
patent: 2742460 (1956-04-01), Murphy et al.
patent: 2798072 (1957-07-01), Pohland
patent: 2850498 (1958-09-01), Pohland
patent: 4764617 (1988-08-01), Masaki et al.
patent: 5030649 (1991-07-01), Vecchietti et al.
patent: 5134238 (1992-07-01), Rossiter et al.
patent: 5646151 (1997-07-01), Kruse et al.
patent: 5804595 (1998-09-01), Portoghese et al.
patent: 256181 (1988-02-01), None
patent: WO 97/46553 (1997-12-01), None
Cignarella et al., Syntheses and κ binding affinity of 1-(pyrrolidin-1-methyl)-2-(N-methyl)-4-[(3,4-dichloro)phenyl]-1,2,3,4-tetrahydroisoquinolin-3(2H)-ones, Eur. J. Med Chem. (1995), 515-520.
Kumar et al., Arylacetamides as Peripherally Restricted Kappa Opioid Receptor Agonists, Bioorganic & Medical Chemistry Letters 10 (2000) 2567-2570.
Singh et al., An Effective Synthesis of Chiral Nonracemic Diamines: Application in Asymmetric Synthesis, Tetrahedron Letters, 39, 1998, 167-170.
O'Brien et al., Practical One-Step Synthesis of Koga's Chiral Bases, Synthesis, 2001, 5, 693-695.
Borisova et al., Aminoamides. III. I-Dialkylamino-3-phenyl-3-acylaminopropanes and I-Dialkylamino-3-phenyl-3-acylaminopropanes, Zhurnal Organicheskoi Khimii, 1969, 5 (2), 284-286.
Moehrle et al., Syntheses of Amino Lactams and Amidines, Archiv der Pharmazie (Weinheim, Germany) 1973, 306 (5), 325-338.
Moehrle et al., Neighboring Group Effects of Aliphatic Amines, Archiv der Pharmazie (Weinheim, Germany) 1973, 306 (3), 209-226.
Curthbertson, Eric, et al., Practical One-Step Synthesis of Koga's Chiral Bases, Dec. 4, 2001, pp. 693-695, Synthesis 2001, No. 5.
Choi Yong-Moon
Kim Yong-Kil
Lee Eun-Ho
Park Chun-Eung
Gibbons, Del Deo, Dolan Griffinger and Vecchione
Nwaonicha Chukwuma
Richter Johann
SK Corporation
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