Drug – bio-affecting and body treating compositions – Designated organic active ingredient containing – Heterocyclic carbon compounds containing a hetero ring...
Reexamination Certificate
2006-11-01
2011-11-08
Moore, Susanna (Department: 1624)
Drug, bio-affecting and body treating compositions
Designated organic active ingredient containing
Heterocyclic carbon compounds containing a hetero ring...
C514S234200, C514S394000, C514S322000, C514S381000, C548S453000, C548S250000, C546S199000, C544S058500, C544S116000
Reexamination Certificate
active
08053431
ABSTRACT:
The use of substituted amides for modulating the activity of 11-hydroxysteroid dehydrogenase type 1 (11HSD1) and the use of these compounds as pharmaceutical compositions, are described. Also a novel class of substituted amides, their use in therapy, pharmaceutical compositions comprising the compounds, as well as their use in the manufacture of medicaments are described. The present compounds are modulators and more specifically inhibitors of the activity of 11HSD1 and may be useful in the treatment, prevention and/or prophylaxis of a range of medical disorders where a decreased intracellular concentration of active glucocorticoid is desirable.
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Andersen Henrik Sune
Ebdrup Soren
Kampen Gita Camilla Tejlgaard
Kilburn John Paul
Dailey Robert S.
High Point Pharmaceuticals, LLC
Moore Susanna
LandOfFree
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