Peripherally selective piperidine opioid antagonists

Drug – bio-affecting and body treating compositions – Designated organic active ingredient containing – Having -c- – wherein x is chalcogen – bonded directly to...

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Details

546231, 546232, 546233, 546234, C07D21126, C07D21128, A61K 31445

Patent

active

052703282

ABSTRACT:
N-alkylamino-3,4,4-substituted piperidines are provided which are useful as peripheral opioid antagonists.

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