Peripherally selective piperidine carboxylate opioid antagonists

Details Peripherally selective piperidine carboxylate opioid antagonists Peripherally selective piperidine carboxylate opioid antagonists

1992-07-17

1993-10-05

Ivy, C. Warren

Drug, bio-affecting and body treating compositions

Designated organic active ingredient containing

Having -c-, wherein x is chalcogen, bonded directly to...

514316, 514318, 514320, 514331, 546187, 546190, 546193, 546207, 546208, 546209, 546231, 546233, 546234, 546235, 546238, 546316, 546318, 546320, 546331, A61K 31445, C07D40112, C07D21132

Patent

active

052505421

ABSTRACT:
3,4,4-trisubstitutedpiperidinyl-N-alkylcarboxylates and intermediates for their preparation are provided. These piperidine-N-alkylcarboxylates are useful as peripheral opioid antagonists.

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