Drug – bio-affecting and body treating compositions – Designated organic active ingredient containing – Peptide containing doai
Patent
1995-06-06
1998-03-10
Johnson, Jerry D.
Drug, bio-affecting and body treating compositions
Designated organic active ingredient containing
Peptide containing doai
530330, 530331, A61K 3806, A61K 3807
Patent
active
057261580
ABSTRACT:
The invention concerns pharmaceutically useful trifluoromethyl ketone substituted di-, tri- and tetra-peptide derivatives of the formulae Ia, Ib, Ic set out hereinafter, and salts thereof, which are inhibitors of human leukocyte elastase. Also described herein are pharmaceutical compositions containing a peptide derivative and processes and intermediates for use in the manufacture of the peptide derivatives.
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Edwards Philip Duke
Schwartz John Anthony
Stein Mark Morris
Trainor Diane Amy
Wildonger Richard Alan
Hohenschutz Liza D.
Johnson Jerry D.
Zeneca Inc.
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