Pentafluorobenzenesulfonamides and analogs

Details Pentafluorobenzenesulfonamides and analogs Pentafluorobenzenesulfonamides and analogs

1999-01-06

2000-09-19

Shah, Mukund J.

Drug, bio-affecting and body treating compositions

Designated organic active ingredient containing

Having -c-, wherein x is chalcogen, bonded directly to...

514415, 514518, 514602, 514604, 5483611, 548469, 558 56, 558 61, 564 90, 564 92, A61K 31415, A01N 4338, C07D23156, C07C30300, C07C30700

Patent

active

061213047

ABSTRACT:
The invention provides methods and compositions relating to novel pentafluorophenylsulfonamide derivatives and analogs and their use as pharmacologically active agents. The compositions find particular use as pharmacological agents in the treatment of disease states, particularly atherosclerosis and hypercholesterolernia, or as lead compounds for the development of such agents. The compositions include compounds of the general formula I: ##STR1##

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