Penicillin esters, salts thereof and methods for their preparati

Details Penicillin esters, salts thereof and methods for their preparati Penicillin esters, salts thereof and methods for their preparati

1975-03-03

1985-11-19

Goldberg, Jerome D.

Drug, bio-affecting and body treating compositions

Plural fermentates of different origin

A61K 3500

Patent

active

045541604

ABSTRACT:
The invention relates to a new series of penicillin esters and salts thereof, to methods of their preparation and to intermediates in the production of the esters of the general formula ##STR1## in which R.sub.1 and R.sub.2 represent an alkyl radical having from 1 to 6 carbon atoms, a cycloalkyl or cycloalkylalkyl radical the cycloalkyl part having from 3 to 10 carbon atoms, or R.sub.1 and R.sub.2 together with the nitrogen atom represent a heterocyclic ring with from 4 to 8 carbon atoms; R.sub.3 represents radicals known from natural, biosynthetic, and semisynthetic penicillins; and pharmaceutically acceptable salts thereof.
The new compounds are efficiently absorbed from the gastrointestinal tract and after the absorption they are rapidly transformed into the corresponding free penicillins and amidinopenicillanic acids, whereby a broad-spectrum infection can be combated.

Affiliated with

Also associated with

Rating

Penicillin esters, salts thereof and methods for their preparati does not yet have a rating. At this time, there are no reviews or comments for this patent.

If you have personal experience with Penicillin esters, salts thereof and methods for their preparati, we encourage you to share that experience with our LandOfFree.com community. Your opinion is very important and Penicillin esters, salts thereof and methods for their preparati will most certainly appreciate the feedback.

Rate now

Comments { 0 }

Profile ID: LFUS-PAI-O-83134