Partial and full agonists of A1 adenosine receptors

Drug – bio-affecting and body treating compositions – Designated organic active ingredient containing – Carbohydrate doai

Reexamination Certificate

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Details

C514S263100, C536S027300, C536S027600, C536S027620, C544S264000, C544S277000

Reexamination Certificate

active

11214706

ABSTRACT:
Disclosed are syntheses suitable for large scale manufacture of novel compounds that are partial and full A1adenosine receptor agonists, useful for treating various disease states, in particular tachycardia and atrial flutter, angina, and myocardial infarction.

REFERENCES:
patent: 5587392 (1996-12-01), Murakami et al.
patent: 6946449 (2005-09-01), Elzein et al.
patent: 7005424 (2006-02-01), Hung et al.
patent: 2003/0216349 (2003-11-01), Belardinelli et al.
patent: 2004/0044225 (2004-03-01), Kanter et al.
patent: 2005/0020532 (2005-01-01), Elzein et al.
patent: 2006/0009417 (2006-01-01), Elzein et al.
Jaworski, J. S. “Nonequilibrium Solvent Polarization in Kinetics of SN2 Reactions,” International Journal of Chemical Kinetics, vol. 35, No. 2, 2003, pp. 61-66.
Van Tilburg et al, “N6,5′—Disubstituted Adenosine Derivatives as Partial Agonists for the Human Adenosine A3Receptor”,J. Med. Chem., Division of Medicinal Chemistry, Leiden/Amsterdam Center for Drug Research, The Netherlands; 1999, vol. 42, pp. 1393-1400.
Robins M.J. et al., “Nucleic Acid Related Compounds. 66. Improved Syntheses of 5′-Chloro-5′-Thionucleosides”, Canadian Journal of Chemistry, National Research Council, Ottawa, Canada, vol. 69, No. 9, 1991, pp. 1468-1474.

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