Packaged stable enema solution or suspension containing 5-aminos

Special receptacle or package – Including ancillary article contacting medium – Gas medium

Patent

Rate now

  [ 0.00 ] – not rated yet Voters 0   Comments 0

Details

514166, B65D 8124, A61K 3160

Patent

active

046642560

ABSTRACT:
A packaged enema solution or suspension consisting essentially of an effective amount of 5-ASA or a pharmaceutically acceptable salt or ester thereof, a chelating agent, an antioxidant and a buffer, the solution or suspension having a pH value of from 4 to 7 and being contained in a plastic bottle under an inert gas, the plastic bottle being packaged in a diffusion-tight light-impervious package in the same inert gas as is present in the bottle.

REFERENCES:
patent: 3044118 (1962-07-01), Bernhardt et al.
patent: 3621892 (1971-11-01), Gillespie
patent: 3937778 (1976-02-01), Tanaka
patent: 4150744 (1979-04-01), Fennimore
patent: 4340550 (1982-07-01), Ho
patent: 4447373 (1984-05-01), Chappell et al.
Khan et al, "An Experiment to Determine the Active Therapeutic Moiety of Sulphasalazine", Lancet, Oct. 29, 1977, pp. 892-895.
Campieri et al, "Treatment of Ulcerative Colitis with High-Dose 5-Amino-Salicyclic Acid Enemas", Lancet, Aug. 8, 1981, pp. 270-271.
Allgayer et al, "Determination of the PK Values of 5-Aminosalicyclic Acid and N-acetylaminosalicyclic Acid and Comparison of the pH Dependent Lipid-Water Partition Coefficients of Sulphasalizine and its Metabolites", Arzneim, Forsch. 35(II), No. 9 (1985), p. 1457-5.
Rhodes, "Medical Treatment of Ulcerative Colitis and Crohn's Disease", Journal of Clinical and Hospital Pharmacy (1983), 8, 219-232.
Bondesen, S. et al, "5-Aminosalicylic Acid Enemas in Patients with Active Ulcertative Colitis", Scand. J. Gastroenterol 19: 677-687 (1984).
Binder, V., "Tropical 5-Aminosalicyclic Acid Versus Prednisolone in Ulcerative Proctosigmoiditis", Digestive Diseases and Sciences, U.S.A., Oct. 3, 1985.
Willoughby, C. et al, "5-Aminosalicyclic Acid (PENTASA) in Enema Form for the Treatment of Active Ulcerative Colitis", Submitted to Scand. J. Gastroenterol.

LandOfFree

Say what you really think

Search LandOfFree.com for the USA inventors and patents. Rate them and share your experience with other people.

Rating

Packaged stable enema solution or suspension containing 5-aminos does not yet have a rating. At this time, there are no reviews or comments for this patent.

If you have personal experience with Packaged stable enema solution or suspension containing 5-aminos, we encourage you to share that experience with our LandOfFree.com community. Your opinion is very important and Packaged stable enema solution or suspension containing 5-aminos will most certainly appreciate the feedback.

Rate now

     

Profile ID: LFUS-PAI-O-1795965

  Search
All data on this website is collected from public sources. Our data reflects the most accurate information available at the time of publication.