Oxazinocarbazoles for the treatment of CNS diseases

Drug – bio-affecting and body treating compositions – In vivo diagnosis or in vivo testing – X-ray contrast imaging agent

Reexamination Certificate

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C424S001810, C544S099000

Reexamination Certificate

active

06932961

ABSTRACT:
The present invention provides isotopically labeled oxazinocarbazole derivatives having a ring connecting position 8 (C-8) and position 9 (N-9), and more specifically, provides compounds of formula (I) wherein R1, R2, R3and R4are described herein.These compounds are useful in the diagnostic analysis of diseases wherein modulation of 5-HT activity is desired.

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