Orally-active elastase inhibitors

Details Orally-active elastase inhibitors Orally-active elastase inhibitors

1995-06-07

1998-02-03

Tsang, Cecilia J.

Drug, bio-affecting and body treating compositions

Designated organic active ingredient containing

Peptide containing doai

514 18, 530330, 530331, A61K 3800

Patent

active

057144702

ABSTRACT:
This invention relates to novel morpholinourea and related derivatives of pentafluoroethyl peptides which are orally active elastase inhibitors. These compounds are useful in the treatment of various inflammatory diseases and emphysema.

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