Organic compounds -- part of the class 532-570 series – Organic compounds – Carbohydrates or derivatives
Patent
1995-06-07
1998-02-24
Wilson, James O.
Organic compounds -- part of the class 532-570 series
Organic compounds
Carbohydrates or derivatives
536 2721, 536 2722, 536 2762, 536 277, C07H 1916
Patent
active
057213569
ABSTRACT:
This invention relates to adenosine kinase inhibitors and to nucleoside analogs, specifically to orally active, substituted 5-aryl analogs having activity as adenosine kinase inhibitors. The invention also relates to the preparation and use of these and other adenosine kinase inhibitors in the treatment of cardiovascular and cerebrovascular diseases, inflammation and other diseases which can be regulated by increasing the local concentration of adenosine.
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Browne Clinton E.
Castellino Angelo J.
Erion Mark D.
Gomez Galeno Jorge E.
Ugarkar Bheemarao G.
Gensia Inc.
Wilson James O.
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