Optically active isomers of quinine and quinidine and their...

Drug – bio-affecting and body treating compositions – Designated organic active ingredient containing – Having -c- – wherein x is chalcogen – bonded directly to...

Reexamination Certificate

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C546S134000, C546S112000, C514S299000

Reexamination Certificate

active

06844355

ABSTRACT:
The present invention provides methods for purifying, identifying and using optically active isomers of quinine and quinidine as well as compositions comprising such optically active isomers. Such optically active isomers having desired actions on cardiac sodium and potassium channel function substantially separable from undesirable effects on GI motility can be useful for more effective therapy of cardiac arrhythmias. Also disclosed are methods for assaying the levels of such isomers present in the biological fluids.

REFERENCES:
patent: 3907806 (1975-09-01), Guenter et al.
patent: 3929795 (1975-12-01), Walter et al.
patent: 0 000 302 (1979-01-01), None
Barhanin et al., (1996)Nature384(6604):78-80.
Bennet et al., (1995)Nature376:683-685.
Busch et al., (1994)Eur J. Pharmacol. 264:33-37.
Catterall, (1992)Physiol. Rev. 72(supp):S15-S48.
Chan et al., (1991)J. Chromatogr. 571:291-297.
Chen et al., (1998)Nature392:293-296.
Coplen et al., (1991)Circulation84:527.
Drabowicz et al., (1984) “Chemical Abstracts”Phosphorus Sulfur16:2676-270 (XP002165239).
Engler et al., (1985)Helv. Chim. Acta. 68:789-800.
Ficker et al., (1998)Circ. Res. 82:386-395.
Gellens et al., (1992)Proc. Natl. Acad. Sci. 89:554-558.
Gutzwiller et al., (1973) “Chemical Abstracts”Helv. Chim. Acta. 79:1494-1503 (XP002165238).
Hartmann et al. (1994)Circ. Res. 75:114-122.
Karle I.L. et al., (1981)Proc. Natl. Acad. Sci. 78:5938-5941.
Karle, J.M. (1997)Antimicrob. Agents Chemother. 41:791-794.
Kiehn et al. (1996)Circulation94:2572-2579.
Krafte et al., (1994)Europ. J. Pharma. 266:245-254.
Li et al. (1996)Circ. Res. 78:689-696.
Sanguinetti et al., (1990)J. Gen. Physiol. 96:195-215.
Sanguinetti et al., (1995)Cell81:299-307.
Sanguinetti et al., (1996)Nature384:80-83.
Spector et al., (1996)J. Gen. Phsyiol. 107:611-619.
Synders et al., (1991)Mol. Pharmacol. 41:322-330.
Trudeau et al., (1995)Science269:92-95.
Van Neuten et al. (1978)Life Sci. 28:453-458.
Wang et al., (1995)Hum. Mol. Genet. 4:1603-1607.
Willius, et al. (1942)Proc. Staff Meet. Mayo Clin. 17:294-296.
International Search Report for International Application PCT/US 00/35213.

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