Oligopeptide prodrugs

Details Oligopeptide prodrugs Oligopeptide prodrugs

1983-06-23

1984-06-12

Phillips, Delbert R.

Chemistry of carbon compounds

Miscellaneous organic carbon compounds

C-metal

C07C10352

Patent

active

044540655

ABSTRACT:
Prodrugs are described whose structures have a oligopeptide chain which is substituted by a nucleophilic chemotherapeutic residue at the .alpha.-position. The products have increased cell membrane permeability and beneficial physico-chemical properties.

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