(o-Acyl-p-N-acylamino-phenyl)-O-phosphoethanolamines

Details (o-Acyl-p-N-acylamino-phenyl)-O-phosphoethanolamines (o-Acyl-p-N-acylamino-phenyl)-O-phosphoethanolamines

1996-10-03

1997-08-26

McKrane, Joseph

Drug, bio-affecting and body treating compositions

Designated organic active ingredient containing

Phosphorus containing other than solely as part of an...

554 41, 558166, A61K 31685, C07F 910

Patent

active

056611382

ABSTRACT:
Novel (o-acyl-p-N-acylamino-phenyl)-O-phosphoethanolamines and pharmaceutically acceptable salts thereof having anti-inflammatory activity, and pharmaceutical compositions containing same are disclosed. Certain novel intermediates are also disclosed.

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Raval, A.A. and Shah, N.M., "Studies in Chalcones and Related Compounds Derived from 2-Hydroxy-5-acetamino-acetophenone. III. Synthesis of 6-Amino-2-methylchromone and 6-Aminoflavone by the Claisen Reaction," J. Org. Chem. (1958) 23:748-749.
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