Novel azolo [1,3] diazepine-5-ol compounds and their uses

Details Novel azolo [1,3] diazepine-5-ol compounds and their uses Novel azolo [1,3] diazepine-5-ol compounds and their uses

1988-02-04

1990-06-19

Brown, Johnnie R.

Organic compounds -- part of the class 532-570 series

Organic compounds

Carbohydrates or derivatives

C07H 19167, C07H 19173, C07H 1702, A61K 3170

Patent

active

049355058

ABSTRACT:
Novel azolo [1,3] diazepine compounds of the formula: ##STR1## wherein R.sup.1 and R.sup.2 are either H or OH and R.sup.1 and R.sup.2 are not the same and X is either CH or N. Such compounds are active as adenosine deaminase inhibitors.

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Elliott et al., Analogs of 8-azaguanosine, Chem Abstracts 85:116642v (1976).
Kanamitsu, Microbial Preduction of Ribosides of Pyrazolo(3,4-d)-Pyrimidines, Chem. Abstracts 80:94260m (1973).
Lichtenthaler et al., Nucleosides 38, The Ribonucleosides of Allopurinol, Chem. Abstracts 95:62573j (1981).
Fryer et al., Quinazolines and 1,4-Benzodiazepines, LXXXVI, The Synthesis of . . . Imidazopyrazolodiazepines, Chem. Abstracts 90:63716 (1978).

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