Nonpeptide endothelin antagonists

Drug – bio-affecting and body treating compositions – Designated organic active ingredient containing – Having -c- – wherein x is chalcogen – bonded directly to...

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514 64, 514 80, 514381, 514382, 514418, 548250, 548251, 548252, 548253, 548405, 548412, 548454, 548484, 548485, 548486, 548490, 548491, 548492, 548503, 548504, 548506, 548507, 548511, A61K 3140, C07D20904

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active

054829607

ABSTRACT:
Novel indole and indoline nonpeptide antagonists of endothelin I are described, as well as novel intermediates used in their preparation, methods for the preparation and pharmaceutical compositions of the same, which are useful in treating elevated levels of endothelin, essential renovascular malignant and pulmonary hypertension, cerebral infarction, cerebral ischemia, congestive heart failure and subarachnoid hemorrhage.

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