Nitroso-N-(.beta.-chloro ethyl)-carbamoyl peptides

Details Nitroso-N-(.beta.-chloro ethyl)-carbamoyl peptides Nitroso-N-(.beta.-chloro ethyl)-carbamoyl peptides

1985-04-19

1990-08-21

Stone, Jacqueline

Drug, bio-affecting and body treating compositions

Designated organic active ingredient containing

Peptide containing doai

530309, 530312, A61K 3702, A61K 3724

Patent

active

049506510

ABSTRACT:
The invention relates to new peptide derivatives of the general Formula I ##STR1## wherein R is a group derived from any oligopeptide by removing a terminal amino group, or--if the oligopeptide comprises a diamino carboxylic acid--the amino group in the .omega.-position, or the terminal and .omega.-amino groups; and

REFERENCES:
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Febs Letters, vol. 44, No. 2 (Aug. 1974), 160-163, Szekerke et al, A New Approach to the Study of the Contribution of Peptide Carriers to Antitumor Activity:Binding of the Peptide Moiety to Human Serum Albumin=Chem. Abstracts (S).
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