Drug – bio-affecting and body treating compositions – Designated organic active ingredient containing – Heterocyclic carbon compounds containing a hetero ring...
Reexamination Certificate
2007-12-07
2010-02-23
Anderson, Rebecca L (Department: 1626)
Drug, bio-affecting and body treating compositions
Designated organic active ingredient containing
Heterocyclic carbon compounds containing a hetero ring...
C514S254010, C514S365000
Reexamination Certificate
active
07666869
ABSTRACT:
The present invention is to provide an aliphatic nitrogen-containing 5-membered ring compound represented by the formula [I]:wherein symbols in the formula have the following meanings;A: —CH2— or —S—,B: CH or N,R1: H, a lower alkyl group, etc.,X: a single bonding arm, —CO—, -Alk-CO—, —COCH2—, -Alk-O—, —O—CH2—, —SO2—, —S—, —COO—, —CON(R3)—, -Alk-CON(R3)—, —CON(R3)CH2—, —NHCH2—, etc.,R3: hydrogen atom or a lower alkyl group,Alk: a lower alkylene group, andR2: (1) a cyclic group which may be substituted,(2) a substituted amino group, etc.,provided that when X is —CO—, then B is N,or a pharmaceutically acceptable salt thereof.
REFERENCES:
patent: 6011155 (2000-01-01), Villhauer
patent: 6107317 (2000-08-01), Villhauer
patent: 6110949 (2000-08-01), Villhauer
patent: 6432969 (2002-08-01), Villhauer
patent: WO 98/19998 (1998-05-01), None
patent: WO 00/34241 (2000-06-01), None
patent: WO 01/96295 (2001-12-01), None
patent: WO 02/051836 (2002-07-01), None
Science (1999), vol. 286, 531-537.
Cancer and Metastasis Reviews (1998), 17(1), 91-106.
Huff, Joel R., “HIV Protease: A Novel Chemotherapeutic Target for AIDS,” Journal of Medicinal Chemistry, vol. 34, No. 8, Aug. 1991, pp. 2305-2314.
Supplementary European Search Report for related application EP 01 97 4716, mailed Apr. 6, 2005.
Augustyns, K., et al., The Unique Properties of Dipeptidyl-peptidase IV (DPP IV / CD 26) and the Therapeutic Potential of DPP IV Inhibitors,Current Medicinal Chemistry, pp. 311-327 (1999).
Arakawa Kenji
Hikota Masataka
Kawanami Saburo
Matsumoto Takeshi
Morimoto Hiroshi
Anderson Rebecca L
Finnegan Henderson Farabow Garrett & Dunner LLP
Mitsubishi Tanabe Pharma Corp.
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