Nitro anthracyclines, process for their preparation and use ther

Details Nitro anthracyclines, process for their preparation and use ther Nitro anthracyclines, process for their preparation and use ther

1986-09-26

1988-06-07

Brown, J. R.

Drug, bio-affecting and body treating compositions

Designated organic active ingredient containing

Carbohydrate doai

536 64, 260365, A61K 3170, C07H 1524

Patent

active

047496932

ABSTRACT:
Anthracycline glycosides of the general formula (A'): ##STR1## wherein R.sub.1 represents a hydrogen atom, a hydroxy group or a methoxy group; one of R.sub.2 and R.sub.3 represents a hydroxy group and the other of R.sub.2 and R.sub.3 represents a nitro group; and R.sub.4 represents a hydrogen atom or a hydroxy group; and their pharmaceutically acceptable salts; have anti-tumor activity.

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