Nicotine receptor ligands

Drug – bio-affecting and body treating compositions – Designated organic active ingredient containing – Heterocyclic carbon compounds containing a hetero ring...

Reexamination Certificate

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Details

C514S210190, C514S233500, C514S256000, C514S307000, C514S320000, C514S337000, C514S422000, C544S062000, C544S151000, C544S153000, C544S333000, C548S525000, C548S950000, C546S139000, C546S144000, C546S148000, C546S196000, C546S282700, C546S284100

Reexamination Certificate

active

06846817

ABSTRACT:
The invention provides nicotine receptor agonists of formula I:wherein R1, x, y, and n have any of the values given in the specification, or a pharmaceutically acceptable salt thereof, as well as pharmaceutical compositions comprising such a compound or salt, methods for preparing such a compound or salt, and methods for modulating (e.g. antagonizing or activating) nicotine receptors with such a compound or salt.

REFERENCES:
patent: 3927023 (1975-12-01), Brown et al.
patent: 4173640 (1979-11-01), Hauck et al.
patent: 4210655 (1980-07-01), Schenker et al.
patent: 4339384 (1982-07-01), Maillard et al.
patent: 4411908 (1983-10-01), Chapleo et al.
patent: 4775675 (1988-10-01), Gyorgydeak et al.
patent: 4940710 (1990-07-01), Sum et al.
patent: 5847159 (1998-12-01), Kai et al.
patent: 613452 (1979-09-01), None
patent: 2408476 (1974-09-01), None
patent: 2408476 (1975-12-01), None
patent: 115142 (1984-08-01), None
patent: 59204190 (1984-11-01), None
patent: 10-175862 (1998-06-01), None
patent: WO 9723216 (1997-07-01), None
patent: 9723216 (1997-07-01), None
patent: 9745424 (1997-12-01), None
patent: WO 0076990 (2000-12-01), None
Schmitt, J.D. et al, “Annual Reports Med. Chem.”, 35, 2000, 41-51.*
Shridhar, D. R.; Sastry, C. V. Reddy; Lal, Kulbhushan; Rao, C. Seshagiri; Taneja, V., Indian Journal of Chemistry, Section B: Organic Chemistry Including Medicinal Chemistry, 18B(3), 254-6 (English) 1979.*
Johansson, Gary; Brisander, Magnus; Sundquist, Staffan; Hacksell, Uli, Chirality, 10(9), 813-820 (English) 1998.*
Document No. 102:185092 Benzofuranylmorpholines. (Kaken Pharmaceutical Co., Ltd., Japan). Jpn. Kokai Tokkyo Koho JP 59204190 A2, Chemical Abstracts.*
Chapleo, C.B., et al., “a-Adrenoreceptor reagents. 2. Effects of modification of the 1,4-benzodioxan ring system on a-adrenoreceptor activity”,Journal of Medicinal Chemistry, 27(5), pp. 570-576, (1984).
Dolby, L.J., et al., “New reactions of 3-vinylindoles”,Tet, vol. 24, No. 21, 6377-6386, (1968).

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